Compound | Agonist pEC50 (IA) | Inverse Agonist (pIC50) | Inhibition (pIC50) | |
---|---|---|---|---|
CB1 | CB2 | GPR55 | S1P1 | |
CP55,940 | 7.1 ± 0.26 (0.3) | 8.3 ± 0.09 (1.0) | 7.6 ± 0.10 | <6.0 |
CP55,667 | 7.0 ± 0.19 (0.3) | 8.2 ± 0.3 (0.8) | 6.8 ± 0.16 | <5.5 |
CP55,244 | 7.3 ± 0.6 (1.0) | 9.2 ± 0.20 (1.0) | 8.3 ± 0.13 | <5.5 |
CP55,243 | <4.5 | 7.2 ± 0.09 (0.3) | 6.9 ± 0.14 | <6.0 |
IA, intrinsic activity.