TABLE 6

Effect of ABT-107 on neurotransmitter uptake activity in rat brain

Assay TypeIC50an
nM
[3H]5-Hydroxytryptamine360 (150–800)6
[3H]Dopamine6900 (2300–11,000)5
[3H]Norepinephrine>10,0005
  • a Values are expressed as means with 95% CI.