TABLE 1
Cellular CYP3A activity
Rates of Product Formation
pmol/20 min/10
5
cells
BEAS-2B cells
0.345 ± 0.0017
WI-38 cells
0.128 ± 0.0004
A549 cells
0.069 ± 0.0002
Mouse lung primary cells
0.197 ± 0.001