Parameter | AC1 | AC2 | AC5 | AC6 | Cardiac AC |
---|---|---|---|---|---|
Km (μM) | 110 ± 29a | 99 ± 22a | 40 ± 5 | 120 ± 42a | 11 ± 2 |
Vmax (pmol · mg–1 · min–1) | 1500 ± 230a | 1200 ± 140a | 3200 ± 400 | 1300 ± 260a | 1010 ± 370 |
Nucleotide, Ki (nM) | |||||
MANT-ITP | 3 | 14 | 1 | 3 | 4 |
MANT-ITPγS | 41a | 120a | 31a | 43a | 8 |
MANT-GTP | 90a | 620a | 55a | 91a | 21 |
MANT-GTPγS | 62a | 360a | 35a | 48a | 23 |
MANT-ATP | 210a | 850a | 200a | 280a | 64 |
MANT-ATPγS | 160 | 380 | 77 | 72 | 67 |
MANT-CTP | 150 | 690 | 150 | 280 | 29 |
MANT-UTP | 46 | 460 | 32 | 71 | 12 |