Parameter | AC1 | AC2 | AC5 | Cardiac AC |
---|---|---|---|---|
Km (μM) | 160 ± 20a | 110 ± 30a | 87 ± 31 | 68 ± 5 |
Vmax (pmol · mg–1 · min–1) | 660 ± 90a | 300 ± 70a | 2400 ± 760 | 1600 ± 160 |
Nucleotide, Ki (nM) | ||||
MANT-ITP | 24 | 65 | 13 | 24 |
MANT-ITPγS | 300a | 450a | 150a | 26 |
MANT-GTP | 1500a | 3700a | 760a | 780 |
MANT-GTPγS | 990a | 1800a | 550a | 340 |
MANT-ATP | 3200a | 5700a | 2000a | 2000 |
MANT-ATPγS | 1400 | 2300 | 1100 | 770 |
MANT-CTP | 3600 | 15,000 | 3600 | 3300 |
MANT-UTP | 1800 | 10,000 | 1000 | 1200 |