Compound | BEI | In Vitro Intrinsic Clbiliarya | ||||
---|---|---|---|---|---|---|
WT | TR– | WT | TR– | |||
% | ml/min/kg | |||||
E2–17βG | 18.4 ± 3.9 | 0.378 ± 0.378 | 17.8 ± 0.4 | 0.363 ± 0.363 | ||
Olmesartan | 14.7 ± 0.5 | 7.05 ± 0.93 | 1.72 ± 0.25 | 0.931 ± 0.167 | ||
Valsartan | 18.9 ± 2.6 | 1.63 ± 1.33 | 3.24 ± 0.51 | 0.406 ± 0.341 | ||
Pravastatin | 43.4 ± 2.3 | 10.7 ± 3.4 | 4.43 ± 0.75 | 1.13 ± 0.33 | ||
Rosuvastatin | 44.9 ± 6.1 | 20.6 ± 3.9 | 46.1 ± 0.4 | 21.2 ± 6.0 | ||
Pitavastatin | 19.9 ± 1.4 | 6.54 ± 3.38 | 34.6 ± 3.1 | 10.4 ± 5.4 |