Compound (+ 5 mM GSH) | Conc. | ATP-Dependent [3H]LTB4 Transport |
---|---|---|
μM | % control | |
[3H]LTB4 (control, 100 nM) | 100 | |
5-Hydroxy-6,8,11,14-eicosatetraenoate | 1 | 86 ± 7 |
12-Hydroxy-5,8,10,14-eicosatetraenoate | 1 | 106 ± 6 |
LTC4 | 1 | 39 ± 4 |
LTD4 | 1 | 67 ± 9 |
S-Decyl GSH | 10 | 26 ± 3 |
Sulindac sulfide | 10 | 26 ± 3 |
Indomethacin | 10 | 32 ± 2 |
Prostaglandin E2 | 10 | 46 ± 5 |
Cholyltaurine | 10 | 39 ± 2 |
Dipyridamole | 10 | 57 ± 3 |
MK571 | 10 | 60 ± 4 |
Montelukast | 10 | 52 ± 5 |
Probenecid | 100 | 73 ± 7 |
Sulfinpyrazone | 100 | 73 ± 7 |