TABLE 1
MCH binding and functional analysis of antagonists
Molecular Mass
MCH1R IC
50
MCH1R K
i
Serotonin
K
i
Da
nM
DABA-821
505
14.0 ± 12.4
39.3 ± 15.0
1155 ± 25
Carboxy-DABA-822
511
35.6 ± 35.9
58.5 ± 22.6
Not tested