Receptor (Expression System) | Radioligand or Agonist | JNJ-17156516 Affinity ± S.E.M. | Dexloxiglumide Affinity ± S.E.M. |
---|---|---|---|
Human CCK1 (CHO) | 125I-CCK-8S | pKI = 7.96 ± 0.11 | pKI = 7.53 ± 0.07 |
Rat CCK1 (CHO) | 125I-CCK-8S | pKI = 8.02 ± 0.11 | pKI = 7.63 ± 0.09 |
Canine CCK1 (CHO) | 125I-CCK-8S | pKI = 7.98 ± 0.04 | pKI = 7.53 ± 0.11 |
Human CCK1 (gallbladder) | [3H]L-364,718 | pKI = 8.22 ± 0.05 | pKI = 7.1 |
Guinea pig CCK1 (gallbladder) | CCK-8S | pKB = 8.00 ± 0.07 | pKB′ = 6.85 ± 0.09 |
Human CCK2 (HEKZFP) | 125I-CCK-8S | pKI = 5.76 ± 0.02 | pKI < 5 |
Rat CCK2 (CHO) | 125I-CCK-8S | pKI = 5.65 ± 0.07 | pKI = 5.23 ± 0.04 |
Canine CCK2 (CHO) | 125I-CCK-8S | pKI = 6.10 ± 0.14 | pKI = 5.56 ± 0.05 |