Compound | 100 nM | 1 μM | 10 μM | 100 μM |
---|---|---|---|---|
Sergliflozin-A | 0.7 ± 3.1 | -3.2 ± 8.3 | -12.7 ± 7.8 | -20.3 ± 18.3 |
Sergliflozin | 3.8 ± 10.5 | -5.0 ± 12.2 | -17.5 ± 8.4 | 22.9 ± 8.7 |
Aglycon of sergliflozin | -13.6 ± 9.6 | 7.5 ± 1.6 | -10.4 ± 11.5 | 31.5 ± 11.9 |
Phlorizin | 19.8 ± 5.5 | 4.0 ± 15.0 | 1.9 ± 14.9 | -1.4 ± 28.9 |
Phloretin | -21.7 ± 17.8 | 19.2 ± 6.0 | 72.2 ± 1.2** | 101.2 ± 1.8** |
↵** p < 0.01 vs. control.