Ki values for sergliflozin-A, sergliflozin, and phlorizin toward human SGLT1 and human SGLT2
Data are presented as means ± S.E.M. (number of experiments).
Compound | Ki toward Human SGLT1 | Ki toward Human SGLT2 |
|---|---|---|
| nM | nM | |
| Sergliflozin-A | 708 ± 50 (5) | 2.39 ± 0.35 (3) |
| Sergliflozin | 7540 ± 402 (8) | 151 ± 17 (3) |
| Phlorizin | 151 ± 8 (5) | 18.6 ± 3.3 (4) |