| | Acetaminophen Sulfate | |
Cliver unbound (nM) | 376 ± 59 | 321 ± 61 | 340 ± 53 |
Clbasolateral (μl/min/g liver) | 142 ± 24 | 117 ± 42 | 111 ± 20 |
Clbile (μl/min/g liver) | 6 ± 1 | 10 ± 3* | 6 ± 1 |
| | 4-Methylumbelliferyl Sulfate | |
Cliver unbound (nM) | 211 ± 55 | 308 ± 166 | 373 ± 91 |
Clbasolateral (μl/min/g liver) | 2036 ± 667 | 1012 ± 354* | 733 ± 235* |
Clbile (μl/min/g liver) | 927 ± 332 | 762 ± 239 | 452 ± 179 |
| | Harmol Sulfate | |
Cliver unbound (nM) | 745 ± 125 | 537 ± 109 | 620 ± 51 |
Clbasolateral (μl/min/g liver) | 411 ± 131 | 296 ± 80 | 229 ± 10 |
Clbile (μl/min/g liver)a | 459 ± 42 | 670 ± 241 | 400 ± 41 |