Peptide | Rat NK1 Receptor (EC50) | Desensitization/Activation Ratio | Human NK1 Receptor (EC50) | Desensitization/Activation Ratio | ||||
---|---|---|---|---|---|---|---|---|
Signal activation | Desensitization | Signal activation | Desensitization | |||||
nM | nM | |||||||
SP | 2.6 | 0.9 | 0.35 | 10.0 | 2.5 | 0.25 | ||
RTKC | 7.3 | 50.6 | 6.93 | 15.3 | 29.2 | 1.93 |