Research ArticleMetabolism, Transport, and Pharmacogenomics
Factors Influencing the CNS Distribution of a Novel PI3K/mTOR Inhibitor GSK2126458: Implications for Overcoming Resistance with Combination Therapy for Melanoma Brain Metastases
Shruthi Vaidhyanathan, Brynna Wilken-Resman, Daniel J Ma, Karen E Parrish, Rajendar K Mittapalli, Brett L Carlson, Jann N. Sarkaria and William F. Elmquist
Journal of Pharmacology and Experimental Therapeutics November 24, 2015, jpet.115.229393; DOI: https://doi.org/10.1124/jpet.115.229393