Research ArticleMetabolism, Transport, and Pharmacogenomics
Brain Distribution and Active Efflux of Three panRAF Inhibitors: Considerations in the Treatment of Melanoma Brain Metastases
Gautham Gampa, Minjee Kim, Afroz S. Mohammad, Karen E. Parrish, Ann C. Mladek, Jann N. Sarkaria and William F. Elmquist
Journal of Pharmacology and Experimental Therapeutics March 2019, 368 (3) 446-461; DOI: https://doi.org/10.1124/jpet.118.253708
Gautham Gampa
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
Minjee Kim
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
Afroz S. Mohammad
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
Karen E. Parrish
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
Ann C. Mladek
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
Jann N. Sarkaria
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
William F. Elmquist
Brain Barriers Research Center, Department of Pharmaceutics, College of Pharmacy, University of Minnesota, Minneapolis, Minnesota (G.G., M.K., A.S.M., K.E.P., W.F.E.); and Radiation Oncology, Mayo Clinic, Rochester, Minnesota (A.C.M., J.N.S.)
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Research ArticleMetabolism, Transport, and Pharmacogenomics
Brain Delivery of panRAF Inhibitors
Gautham Gampa, Minjee Kim, Afroz S. Mohammad, Karen E. Parrish, Ann C. Mladek, Jann N. Sarkaria and William F. Elmquist
Journal of Pharmacology and Experimental Therapeutics March 1, 2019, 368 (3) 446-461; DOI: https://doi.org/10.1124/jpet.118.253708
Research ArticleMetabolism, Transport, and Pharmacogenomics
Brain Delivery of panRAF Inhibitors
Gautham Gampa, Minjee Kim, Afroz S. Mohammad, Karen E. Parrish, Ann C. Mladek, Jann N. Sarkaria and William F. Elmquist
Journal of Pharmacology and Experimental Therapeutics March 1, 2019, 368 (3) 446-461; DOI: https://doi.org/10.1124/jpet.118.253708
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