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Discovery of 1-((6-Aminopyridin-3-yl)Methyl)-3-(4-Bromophenyl)Urea as a Potent, Irreversible Myeloperoxidase Inhibitor
Martin L. Marro, Andrew W. Patterson, Lac Lee, Lin Deng, Aimee Reynolds, Xianglin Ren, Laura Axford, Anup Patnaik, Micah Hollis-Symynkywicz, Nigel Casson, Dominique Custeau, Lisa Ames, Sally Loi, Lihe Zhang, Toshiyuki Honda, Jutta Blank, Tyler J. Harrison, Julien P. N. Papillon, Lawrence G. Hamann, Jovita Marcinkeviciene and Jean B. Regard
Journal of Pharmacology and Experimental Therapeutics October 2018, 367 (1) 147-154; DOI: https://doi.org/10.1124/jpet.118.248435