Research ArticleMETABOLISM, TRANSPORT, AND PHARMACOGENOMICS
CYP2C75-Involved Autoinduction of Metabolism in Rhesus Monkeys of Methyl 3-Chloro-3′-fluoro-4′-{(1R)-1-[({1-[(trifluoroacetyl)amino]cyclopropyl}carbonyl)amino]ethyl}-1,1′-biphenyl-2-carboxylate (MK-0686), a Bradykinin B1 Receptor Antagonist
Cuyue Tang, Brian A. Carr, Frédéric Poignant, Bennett Ma, Stacey L. Polsky-Fisher, Yuhsin Kuo, Kristie Strong-Basalyga, Alisha Norcross, Karen Richards, Roy Eisenhandler, Edward J. Carlini, Christina Ng Di Marco, Scott D. Kuduk, Nathan X. Yu, Conrad E. Raab, Tom Rushmore, Clay B. Frederick, Mark G. Bock and Thomayant Prueksaritanont
Journal of Pharmacology and Experimental Therapeutics June 2008, 325 (3) 935-946; DOI: https://doi.org/10.1124/jpet.107.136044
Cuyue Tang
Brian A. Carr
Frédéric Poignant
Bennett Ma
Stacey L. Polsky-Fisher
Yuhsin Kuo
Kristie Strong-Basalyga
Alisha Norcross
Karen Richards
Roy Eisenhandler
Edward J. Carlini
Christina Ng Di Marco
Scott D. Kuduk
Nathan X. Yu
Conrad E. Raab
Tom Rushmore
Clay B. Frederick
Mark G. Bock
Thomayant Prueksaritanont
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Research ArticleMETABOLISM, TRANSPORT, AND PHARMACOGENOMICS
CYP2C75-Involved Autoinduction of Metabolism in Rhesus Monkeys of Methyl 3-Chloro-3′-fluoro-4′-{(1R)-1-[({1-[(trifluoroacetyl)amino]cyclopropyl}carbonyl)amino]ethyl}-1,1′-biphenyl-2-carboxylate (MK-0686), a Bradykinin B1 Receptor Antagonist
Cuyue Tang, Brian A. Carr, Frédéric Poignant, Bennett Ma, Stacey L. Polsky-Fisher, Yuhsin Kuo, Kristie Strong-Basalyga, Alisha Norcross, Karen Richards, Roy Eisenhandler, Edward J. Carlini, Christina Ng Di Marco, Scott D. Kuduk, Nathan X. Yu, Conrad E. Raab, Tom Rushmore, Clay B. Frederick, Mark G. Bock and Thomayant Prueksaritanont
Journal of Pharmacology and Experimental Therapeutics June 1, 2008, 325 (3) 935-946; DOI: https://doi.org/10.1124/jpet.107.136044
Research ArticleMETABOLISM, TRANSPORT, AND PHARMACOGENOMICS
CYP2C75-Involved Autoinduction of Metabolism in Rhesus Monkeys of Methyl 3-Chloro-3′-fluoro-4′-{(1R)-1-[({1-[(trifluoroacetyl)amino]cyclopropyl}carbonyl)amino]ethyl}-1,1′-biphenyl-2-carboxylate (MK-0686), a Bradykinin B1 Receptor Antagonist
Cuyue Tang, Brian A. Carr, Frédéric Poignant, Bennett Ma, Stacey L. Polsky-Fisher, Yuhsin Kuo, Kristie Strong-Basalyga, Alisha Norcross, Karen Richards, Roy Eisenhandler, Edward J. Carlini, Christina Ng Di Marco, Scott D. Kuduk, Nathan X. Yu, Conrad E. Raab, Tom Rushmore, Clay B. Frederick, Mark G. Bock and Thomayant Prueksaritanont
Journal of Pharmacology and Experimental Therapeutics June 1, 2008, 325 (3) 935-946; DOI: https://doi.org/10.1124/jpet.107.136044
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