| % | |
nM
| |
Adenosine A1 | <10 | CPA | 0.88 | Rat cerebral cortex |
Adenosine A2A | <10 | NECA | 4.5 | Rat striatum |
Adrenaline α1 (nonselective) | <10 | Prazosin | 0.42 | Rat cerebral cortex |
Adrenaline α2 (nonselective) | <10 | Yohimbine | 66 | Rat cerebral cortex |
Adrenaline β1 | <10 | Atenolol | 1320 | Rat heart |
Angiotensin (AT1) | <10 | Saralasin | 1.6 | Rat lung |
Angiotensin (AT2) | <10 | Saralasin | 2.8 | Bovine cerebellum |
ANP | <10 | ANP | 0.11 | Guinea pig cerebellum |
BDZ (central) | <10 | Diazepam | 25 | Rat cerebral cortex |
Bradykinin (B2) | <10 | NPC567 | 6.1 | Human recombinant (CHO cell) |
Cholecystokinin (CCK1) | <10 | Devazepide | 0.62 | Human recombinant (NIH3T3 cell) |
CRF1 | <10 | CRF | 6.3 | Rat pituitary gland |
Dopamine (D1) | <10 | SCH23390 | 0.92 | Rat striatum |
Dopamine (D2) | <10 | (+)Butaclamol | 3.9 | Rat striatum |
Endothelin A | <10 | Endothelin-1 | 0.42 | a-10 cells |
GABA (nonselective) | <10 | GABA | 29 | Rat cerebral cortex |
NMDA | <10 | CGS19755 | 1380 | Rat cerebral cortex |
PDGF | <10 | PDGF BB | 0.58 | Balb/c 3T3 cells |
IL-1β | <10 | IL-1β | 0.039 | Balb/c 3T3 cells |
TNF-α | <10 | TNF-α | 0.19 | U937 cells |
Histamine (H1 central) | <10 | Pyrilamine | 1.2 | Guinea pig cerebellum |
Insulin | <10 | Insulin | 12 | Rat liver |
Muscarine (nonselective) | 12 | Atropine | 0.65 | Rat cerebral cortex |
Neurokinin (NK1) | <10 | [Sar9,Met(O2)11]-SP | 1.5 | U-373MG cells |
NPY (nonselective) | 12 | NPY | 0.91 | Rat cerebral cortex |
Nicotine (neuronal) | <10 | Nicotine | 28 | Rat cerebral cortex |
Opiate (nonselective) | 15 | Naloxone | 1.6 | Rat cerebral cortex |
PAF | <10 | WEB2086 | 3.9 | Rabbit platelet |
PCP | <10 | MK801 | 2.4 | Rat cerebral cortex |
5-HT (nonselective) | <10 | Serotonin | 1.9 | Rat cerebral cortex |
5-HT1B | <10 | Serotonin | 20 | Rat cerebral cortex |
5-HT2A | <10 | Ketanserin | 1.7 | Rat cerebral cortex |
σ (nonselective) | <10 | Haloperidol | 72 | Rat cerebral cortex |
Glucocorticoid | <10 | Dexamethasone | 117 | L-929 cells (cytosol) |
VIP1 | 14 | VIP | 1.6 | HT-29 cells |
L-type Ca2+ channel | <10 | Nitrendipine | 16 | A7r5 cells |
COX-1 | <10 | Diclofenac | 85 | Rat seminal vesicle |
COX-2 | 11 | NS398 | 5200 | Sheep placenta |
Inducible NOS | <10 | l-NMMA | 466,000 | RAW264-7 cells |
Constitutive NOS | 11 | l-NMMA | 280 | HUVEC |
Phosphodiesterase I | <10 | 8-Methoxy-IBMX | 1800 | Bovine brain |
Phosphodiesterase III | <10 | Milrinone | 220 | Guinea pig heart |
Phosphodiesterase IV | <10 | Rolipram | 200 | U-937 cells |
Phosphodiesterase V | <10 | Dipyridamole | 230 | Human platelets |
Aldose reductase | <10 | ICI-128,436 | 4.1 | Bovine lens |
ACE | <10 | Captopril | 1.5 | HUVEC |
Caspase-3
| <10
| DEVD-CHO
| 230
| U937 cells
|