Table of Contents

October 1994; 271 (1)

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- M Gekle,
- S Mildenberger,
- R Freudinger,
- and S Silbernagl
The mycotoxin ochratoxin-A impairs protein uptake in cells derived from the proximal tubule of the kidney (opossum kidney cells).
J Pharmacol Exp Ther October 1994 271:1-6
- Abstract
- Full Text (PDF)
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- U Scheurer,
- E Drack,
- and F Halter
Substance P activates rat colonic motility via excitatory and inhibitory neural pathways and direct action on muscles.
J Pharmacol Exp Ther October 1994 271:7-13
- Abstract
- Full Text (PDF)
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- K Niiya,
- S Uchida,
- T Tsuji,
- and R A Olsson
Glibenclamide reduces the coronary vasoactivity of adenosine receptor agonists.
J Pharmacol Exp Ther October 1994 271:14-19
- Abstract
- Full Text (PDF)
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- M Oshita,
- Y Takei,
- S Kawano,
- H Fusamoto,
- and T Kamada
Protective effect of ebselen on constrictive hepatic vasculature: prevention of alcohol-induced effects on portal pressure in perfused livers.
J Pharmacol Exp Ther October 1994 271:20-24
- Abstract
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- S D Donevan,
- S Yamaguchi,
- and M A Rogawski
Non-N-methyl-D-aspartate receptor antagonism by 3-N-substituted 2,3-benzodiazepines: relationship to anticonvulsant activity.
J Pharmacol Exp Ther October 1994 271:25-29
- Abstract
- Full Text (PDF)
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- G A Skeen,
- H S White,
- and R E Twyman
The dihydropyridine nitrendipine reduces N-methyl-D-aspartate (NMDA)-evoked currents of rodent cortical neurons through a direct interaction with the NMDA receptor-associated ion channel.
J Pharmacol Exp Ther October 1994 271:30-38
- Abstract
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- M B Parrish,
- K D Rainsford,
- D M Johnson,
- and E E Daniel
NK1 receptors mediated release of 6-keto-PGF1 alpha from the ex vivo perfused canine ileum.
J Pharmacol Exp Ther October 1994 271:39-47
- Abstract
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- K L Preston and
- G E Bigelow
Drug discrimination assessment of agonist-antagonist opioids in humans: a three-choice saline-hydromorphone-butorphanol procedure.
J Pharmacol Exp Ther October 1994 271:48-60
- Abstract
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- T D Hexum,
- J Zheng,
- and J Zhu
Neuropeptide Y inhibition of nicotinic receptor-mediated chromaffin cell secretion.
J Pharmacol Exp Ther October 1994 271:61-66
- Abstract
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- L J Chandler,
- N J Guzman,
- C Sumners,
- and F T Crews
Magnesium and zinc potentiate ethanol inhibition of N-methyl-D-aspartate-stimulated nitric oxide synthase in cortical neurons.
J Pharmacol Exp Ther October 1994 271:67-75
- Abstract
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- K A Sluka,
- W D Willis,
- and K N Westlund
Inflammation-induced release of excitatory amino acids is prevented by spinal administration of a GABAA but not by a GABAB receptor antagonist in rats.
J Pharmacol Exp Ther October 1994 271:76-82
- Abstract
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- S Prisco,
- S Pagannone,
- and E Esposito
Serotonin-dopamine interaction in the rat ventral tegmental area: an electrophysiological study in vivo.
J Pharmacol Exp Ther October 1994 271:83-90
- Abstract
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- L Perrier,
- M Bourrié,
- E Marti,
- C Tronquet,
- D Massé,
- Y Berger,
- J Magdalou,
- and G Fabre
In vitro N-glucuronidation of SB 47436 (BMS 186295), a new AT1 nonpeptide angiotensin II receptor antagonist, by rat, monkey and human hepatic microsomal fractions.
J Pharmacol Exp Ther October 1994 271:91-99
- Abstract
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- K Nomura,
- N Maeda,
- T Yoshino,
- and I Yamaguchi
A mechanism of 5-HT3 receptor mediation is involved etiologically in the psychological stress lesion the stomach of the mouse.
J Pharmacol Exp Ther October 1994 271:100-106
- Abstract
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- C Dominice,
- M N Dufour,
- N Patino,
- O Manzoni,
- E Grazzini,
- P Jouin,
- and G Guillon
Dual effects of nordidemnin on WRK1 cells: inhibition of phosphoinositide metabolism and cell proliferation.
J Pharmacol Exp Ther October 1994 271:107-117
- Abstract
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- L J Murphey and
- G D Olsen
Diffusion of morphine-6-beta-D-glucuronide into the neonatal guinea pig brain during drug-induced respiratory depression.
J Pharmacol Exp Ther October 1994 271:118-124
- Abstract
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- A C Collins,
- Y Luo,
- S Selvaag,
- and M J Marks
Sensitivity to nicotine and brain nicotinic receptors are altered by chronic nicotine and mecamylamine infusion.
J Pharmacol Exp Ther October 1994 271:125-133
- Abstract
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- M Buerke,
- A S Weyrich,
- T Murohara,
- C Queen,
- C K Klingbeil,
- M S Co,
- and A M Lefer
Humanized monoclonal antibody DREG-200 directed against I-selectin protects in feline myocardial reperfusion injury.
J Pharmacol Exp Ther October 1994 271:134-142
- Abstract
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- C S Aulakh,
- P Mazzola-Pomietto,
- J L Hill,
- and D L Murphy
Role of various 5-HT receptor subtypes in mediating neuroendocrine effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM) in rats.
J Pharmacol Exp Ther October 1994 271:143-148
- Abstract
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- P Cuq,
- R Magous,
- and J P Bali
Pharmacological coupling and functional role for the muscarinic receptor subtypes in isolated cells from the circular smooth muscle of the rabbit cecum.
J Pharmacol Exp Ther October 1994 271:149-155
- Abstract
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- T Yamamoto,
- N Shimoyama,
- H Asano,
- and T Mizuguchi
Analysis of the role of endothelin-A and endothelin-B receptors on nociceptive information transmission in the spinal cord with FR139317, an endothelin-A receptor antagonist, and sarafotoxin S6c, an endothelin-B receptor agonist.
J Pharmacol Exp Ther October 1994 271:156-163
- Abstract
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- D A Finn and
- K W Gee
The estrus cycle, sensitivity to convulsants and the anticonvulsant effect of a neuroactive steroid.
J Pharmacol Exp Ther October 1994 271:164-170
- Abstract
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- H Vidrio
Potentiation of cardiovascular responses to hydralazine by diverse hydrazine derivatives.
J Pharmacol Exp Ther October 1994 271:171-175
- Abstract
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- A M Gillis,
- M Choi,
- H J Mathison,
- and H G Parsons
Influence of dietary fat on the pharmacodynamics of quinidine, procainamide and tocainide in isolated perfused rabbit hearts.
J Pharmacol Exp Ther October 1994 271:176-183
- Abstract
- Full Text (PDF)
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- J S Pasnani and
- G R Ferrier
Pro- and antiarrhythmic effects of d-sotalol and dl-sotalol in an isolated tissue model of ischemia and reperfusion.
J Pharmacol Exp Ther October 1994 271:184-192
- Abstract
- Full Text (PDF)
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- H Defacque,
- J Dornand,
- T Commes,
- S Cabane,
- C Sevilla,
- and J Marti
Different combinations of retinoids and vitamin D3 analogs efficiently promote growth inhibition and differentiation of myelomonocytic leukemia cell lines.
J Pharmacol Exp Ther October 1994 271:193-199
- Abstract
- Full Text (PDF)
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- R B Stewart,
- G A Lemaire,
- J D Roache,
- and R A Meisch
Establishing benzodiazepines as oral reinforcers: midazolam and diazepam self-administration in rhesus monkeys.
J Pharmacol Exp Ther October 1994 271:200-211
- Abstract
- Full Text (PDF)
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- G M Gonzalez-Alvear and
- L L Werling
Regulation of [3H]dopamine release from rat striatal slices by sigma receptor ligands.
J Pharmacol Exp Ther October 1994 271:212-219
- Abstract
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- S Desai,
- T Hadlock,
- C Messam,
- R Chafetz,
- and G Strichartz
Ionization and adsorption of a series of local anesthetics in detergent micelles: studies of drug fluorescence.
J Pharmacol Exp Ther October 1994 271:220-228
- Abstract
- Full Text (PDF)
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- S R Doctrow,
- S M Abelleira,
- L A Curry,
- R Heller-Harrison,
- J W Kozarich,
- B Malfroy,
- L A McCarroll,
- K G Morgan,
- A R Morrow,
- and G F Musso
The bradykinin analog RMP-7 increases intracellular free calcium levels in rat brain microvascular endothelial cells.
J Pharmacol Exp Ther October 1994 271:229-237
- Abstract
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- Z Y Friedman
The antitumor agent tamoxifen inhibits breakdown of polyphosphoinositides in GH4C1 cells.
J Pharmacol Exp Ther October 1994 271:238-245
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- J M O'Donnell,
- S Frith,
- and J Wilkins
Involvement of beta-1 and beta-2 adrenergic receptors in the antidepressant-like effects of centrally administered isoproterenol.
J Pharmacol Exp Ther October 1994 271:246-254
- Abstract
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- G E Torres,
- I L Holt,
- and R Andrade
Antagonists of 5-HT4 receptor-mediated responses in adult hippocampal neurons.
J Pharmacol Exp Ther October 1994 271:255-261
- Abstract
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- P Fan,
- S Visentin,
- and F F Weight
Effects of cocaine on the serotonin-induced inward current in rat nodose ganglion neurons.
J Pharmacol Exp Ther October 1994 271:262-266
- Abstract
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- C Labbé-Jullié,
- S Deschaintres,
- D Gully,
- G Le Fur,
- and P Kitabgi
Effect of the nonpeptide neurotensin antagonist, SR 48692, and two enantiomeric analogs, SR 48527 and SR 49711, on neurotensin binding and contractile responses in guinea pig ileum and colon.
J Pharmacol Exp Ther October 1994 271:267-276
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- T Shibamoto,
- S Chakder,
- and S Rattan
Role of hypogastric nerve activity in opossum internal anal sphincter function: influence of surgical and chemical denervation.
J Pharmacol Exp Ther October 1994 271:277-284
- Abstract
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- H W Broening,
- L Bacon,
- and W Slikker, Jr
Age modulates the long-term but not the acute effects of the serotonergic neurotoxicant 3,4-methylenedioxymethamphetamine.
J Pharmacol Exp Ther October 1994 271:285-293
- Abstract
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- P Bauco and
- R A Wise
Potentiation of lateral hypothalamic and midline mesencephalic brain stimulation reinforcement by nicotine: examination of repeated treatment.
J Pharmacol Exp Ther October 1994 271:294-301
- Abstract
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- T Sawanobori,
- H Adaniya,
- T Namiki,
- and M Hiraoka
Rate-dependent effects of sematilide on action potential duration in isolated guinea pig ventricular myocytes.
J Pharmacol Exp Ther October 1994 271:302-310
- Abstract
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- J Mattana,
- N Gibbons,
- and P C Singhal
Cocaine interacts with macrophages to modulate mesangial cell proliferation.
J Pharmacol Exp Ther October 1994 271:311-318
- Abstract
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- Y Q Xu,
- W J Crumb, Jr,
- and C W Clarkson
Cocaethylene, a metabolite of cocaine and ethanol, is a potent blocker of cardiac sodium channels.
J Pharmacol Exp Ther October 1994 271:319-325
- Abstract
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- F Zhang and
- A H Morice
Effect of levcromakalim on hypoxia-, KCl- and prostaglandin F2 alpha-induced contractions in isolated rat pulmonary artery.
J Pharmacol Exp Ther October 1994 271:326-333
- Abstract
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- S S Osmanovic and
- S A Shefner
Ethanol enhances inward rectification in rat locus ceruleus neurons by increasing the extracellular potassium concentration.
J Pharmacol Exp Ther October 1994 271:334-342
- Abstract
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- I Krisch,
- B Bole-Vunduk,
- M Pepelnak,
- B Lavric,
- A Ocvirk,
- M V Budihna,
- and D Sket
Pharmacological studies with two new ergoline derivatives, the potential antipsychotics LEK-8829 and LEK-8841.
J Pharmacol Exp Ther October 1994 271:343-352
- Abstract
- Full Text (PDF)
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- J D Brioni,
- A B O'Neill,
- D J Kim,
- M J Buckley,
- M W Decker,
- and S P Arneric
Anxiolytic-like effects of the novel cholinergic channel activator ABT-418.
J Pharmacol Exp Ther October 1994 271:353-361
- Abstract
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- X Xu,
- T D Tsai,
- J Wang,
- E W Lee,
- and K S Lee
Modulation of three types of K+ currents in canine coronary artery smooth muscle cells by NS-004, or 1-(2'-hydroxy-5'-chlorophenyl)-5-trifluoromethyl-2(3H) benzimidazolone.
J Pharmacol Exp Ther October 1994 271:362-369
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- H Shimamura,
- H Suzuki,
- M Hanano,
- A Suzuki,
- O Tagaya,
- T Horie,
- and Y Sugiyama
Multiple systems for the biliary excretion of organic anions in rats: liquiritigenin conjugates as model compounds.
J Pharmacol Exp Ther October 1994 271:370-378
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- H Miyahara,
- Y Kawai,
- and T Ohhashi
5-Hydroxytryptamine-2 and -4 receptors located on bovine isolated mesenteric lymphatics.
J Pharmacol Exp Ther October 1994 271:379-385
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- H P Voss,
- S Shukrula,
- T S Wu,
- D Donnell,
- and A Bast
A functional beta-2 adrenoceptor-mediated chronotropic response in isolated guinea pig heart tissue: selectivity of the potent beta-2 adrenoceptor agonist TA 2005.
J Pharmacol Exp Ther October 1994 271:386-389
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- G C Smith,
- R A Coleman,
- and J C McGrath
Characterization of dilator prostanoid receptors in the fetal rabbit ductus arteriosus.
J Pharmacol Exp Ther October 1994 271:390-396
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- F Ueda,
- Y Kameda,
- O Yamamoto,
- and Y Shibata
Beta-adrenergic regulation of gap-junctional intercellular communication in cultured rabbit gastric epithelial cells.
J Pharmacol Exp Ther October 1994 271:397-402
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- F X Beck,
- A Ohno,
- A Dörge,
- and K Thurau
Loop diuretics affect transcellular electrolyte transport in cells of the distal convoluted tubule.
J Pharmacol Exp Ther October 1994 271:403-407
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- J F Ewing,
- V S Raju,
- and M D Maines
Induction of heart heme oxygenase-1 (HSP32) by hyperthermia: possible role in stress-mediated elevation of cyclic 3':5'-guanosine monophosphate.
J Pharmacol Exp Ther October 1994 271:408-414
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- L A Erickson,
- P D Bonin,
- D G Wishka,
- J Morris,
- R J Dalga,
- D J Williams,
- G J Wilson,
- J L Hoover,
- C A Simmons,
- and S J Humphrey
In vitro and in vivo inhibition of rat vascular smooth muscle cell migration and proliferation by a 2-aminochromone U-86983.
J Pharmacol Exp Ther October 1994 271:415-421
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- P Butkerait,
- H Y Wang,
- and E Friedman
Increases in guanine nucleotide binding to striatal G proteins is associated with dopamine receptor supersensitivity.
J Pharmacol Exp Ther October 1994 271:422-428
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- C P Sung,
- A J Arleth,
- B L Storer,
- and E H Ohlstein
Angiotensin type 1 receptors mediate smooth muscle proliferation and endothelin biosynthesis in rat vascular smooth muscle.
J Pharmacol Exp Ther October 1994 271:429-437
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- P Liu,
- S L Vonderfecht,
- G M McGuire,
- M A Fisher,
- A Farhood,
- and H Jaeschke
The 21-aminosteroid tirilazad mesylate protects against endotoxin shock and acute liver failure in rats.
J Pharmacol Exp Ther October 1994 271:438-445
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- D J Crutchley,
- L B Conanan,
- and B G Que
Effects of prostacyclin analogs on the synthesis of tissue factor, tumor necrosis factor-alpha and interleukin-1 beta in human monocytic THP-1 cells.
J Pharmacol Exp Ther October 1994 271:446-451
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- X Ligneau,
- M Garbarg,
- M L Vizuete,
- J Diaz,
- K Purand,
- H Stark,
- W Schunack,
- and J C Schwartz
[125I]iodoproxyfan, a new antagonist to label and visualize cerebral histamine H3 receptors.
J Pharmacol Exp Ther October 1994 271:452-459
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- K M Merchant,
- D J Dobie,
- F M Filloux,
- M Totzke,
- M Aravagiri,
- and D M Dorsa
Effects of chronic haloperidol and clozapine treatment on neurotensin and c-fos mRNA in rat neostriatal subregions.
J Pharmacol Exp Ther October 1994 271:460-471
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- J P Wagner,
- F J Seidler,
- S E Lappi,
- E C McCook,
- and T A Slotkin
Role of thyroid status in the ontogeny of adrenergic cell signaling in rat brain: beta receptors, adenylate cyclase, ornithine decarboxylase and c-fos protooncogene expression.
J Pharmacol Exp Ther October 1994 271:472-483
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- D W Bonhaus,
- D N Loury,
- L B Jakeman,
- S A Hsu,
- Z P To,
- E Leung,
- K D Zeitung,
- R M Eglen,
- and E H Wong
[3H]RS-23597-190, a potent 5-hydroxytryptamine4 antagonist labels sigma-1 but not sigma-2 binding sites in guinea pig brain.
J Pharmacol Exp Ther October 1994 271:484-493
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- M Alkondon,
- S Reinhardt,
- C Lobron,
- B Hermsen,
- A Maelicke,
- and E X Albuquerque
Diversity of nicotinic acetylcholine receptors in rat hippocampal neurons. II. The rundown and inward rectification of agonist-elicited whole-cell currents and identification of receptor subunits by in situ hybridization.
J Pharmacol Exp Ther October 1994 271:494-506
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- D Gelperin,
- D Mann,
- J del Valle,
- and J W Wiley
Bradykinin (Bk) increases cytosolic calcium in cultured rat myenteric neurons via Bk-2 type receptors coupled to mobilization of extracellular and intracellular sources of calcium: evidence that calcium influx is prostaglandin dependent.
J Pharmacol Exp Ther October 1994 271:507-514
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- M E Fitzsimmons,
- R B Baggs,
- and M W Anders
Nephrotoxicity and hepatotoxicity of 5,6-dichloro-4-thia-5-hexenoic acid: evidence for fatty acid beta-oxidation-dependent bioactivation.
J Pharmacol Exp Ther October 1994 271:515-523
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- Z H Meng and
- M S Dar
Intrastriatal Ro15-4513 functionally antagonizes ethanol-induced motor incoordination and striatal adenosinergic modulation of ethanol-induced motor incoordination in rats.
J Pharmacol Exp Ther October 1994 271:524-534
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- J Neumann,
- P Bokník,
- S Herzig,
- W Schmitz,
- H Scholz,
- K Wiechen,
- and N Zimmermann
Biochemical and electrophysiological mechanisms of the positive inotropic effect of calyculin A, a protein phosphatase inhibitor.
J Pharmacol Exp Ther October 1994 271:535-541
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- M K Sapru,
- I Diamond,
- and A S Gordon
Adenosine receptors mediate cellular adaptation to ethanol in NG108-15 cells.
J Pharmacol Exp Ther October 1994 271:542-548
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- K E Thummel,
- D D Shen,
- T D Podoll,
- K L Kunze,
- W F Trager,
- P S Hartwell,
- V A Raisys,
- C L Marsh,
- J P McVicar,
- and D M Barr
Use of midazolam as a human cytochrome P450 3A probe: I. In vitro-in vivo correlations in liver transplant patients.
J Pharmacol Exp Ther October 1994 271:549-556
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- K E Thummel,
- D D Shen,
- T D Podoll,
- K L Kunze,
- W F Trager,
- C E Bacchi,
- C L Marsh,
- J P McVicar,
- D M Barr,
- and J D Perkins
Use of midazolam as a human cytochrome P450 3A probe: II. Characterization of inter- and intraindividual hepatic CYP3A variability after liver transplantation.
J Pharmacol Exp Ther October 1994 271:557-566
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- Y W Liu,
- Y Asaoka,
- H Suzuki,
- T Yoshimoto,
- S Yamamoto,
- and W C Chang
Induction of 12-lipoxygenase expression by epidermal growth factor is mediated by protein kinase C in A431 cells.
J Pharmacol Exp Ther October 1994 271:567-573
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- M Satoh,
- T Sakai,
- I Sano,
- K Fujikura,
- H Koyama,
- K Ohshima,
- Z Itoh,
- and S Omura
EM574, an erythromycin derivative, is a potent motilin receptor agonist in human gastric antrum.
J Pharmacol Exp Ther October 1994 271:574-579
- Abstract
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Current Issue

November 2009, 331 (2)

The mycotoxin ochratoxin-A impairs protein uptake in cells derived from the proximal tubule of the kidney (opossum kidney cells).

Substance P activates rat colonic motility via excitatory and inhibitory neural pathways and direct action on muscles.

Glibenclamide reduces the coronary vasoactivity of adenosine receptor agonists.

Protective effect of ebselen on constrictive hepatic vasculature: prevention of alcohol-induced effects on portal pressure in perfused livers.

Non-N-methyl-D-aspartate receptor antagonism by 3-N-substituted 2,3-benzodiazepines: relationship to anticonvulsant activity.

The dihydropyridine nitrendipine reduces N-methyl-D-aspartate (NMDA)-evoked currents of rodent cortical neurons through a direct interaction with the NMDA receptor-associated ion channel.

NK1 receptors mediated release of 6-keto-PGF1 alpha from the ex vivo perfused canine ileum.

Drug discrimination assessment of agonist-antagonist opioids in humans: a three-choice saline-hydromorphone-butorphanol procedure.

Neuropeptide Y inhibition of nicotinic receptor-mediated chromaffin cell secretion.

Magnesium and zinc potentiate ethanol inhibition of N-methyl-D-aspartate-stimulated nitric oxide synthase in cortical neurons.

Inflammation-induced release of excitatory amino acids is prevented by spinal administration of a GABAA but not by a GABAB receptor antagonist in rats.

Serotonin-dopamine interaction in the rat ventral tegmental area: an electrophysiological study in vivo.

In vitro N-glucuronidation of SB 47436 (BMS 186295), a new AT1 nonpeptide angiotensin II receptor antagonist, by rat, monkey and human hepatic microsomal fractions.

A mechanism of 5-HT3 receptor mediation is involved etiologically in the psychological stress lesion the stomach of the mouse.

Dual effects of nordidemnin on WRK1 cells: inhibition of phosphoinositide metabolism and cell proliferation.

Diffusion of morphine-6-beta-D-glucuronide into the neonatal guinea pig brain during drug-induced respiratory depression.

Sensitivity to nicotine and brain nicotinic receptors are altered by chronic nicotine and mecamylamine infusion.

Humanized monoclonal antibody DREG-200 directed against I-selectin protects in feline myocardial reperfusion injury.

Role of various 5-HT receptor subtypes in mediating neuroendocrine effects of 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane (DOM) in rats.

Pharmacological coupling and functional role for the muscarinic receptor subtypes in isolated cells from the circular smooth muscle of the rabbit cecum.

Analysis of the role of endothelin-A and endothelin-B receptors on nociceptive information transmission in the spinal cord with FR139317, an endothelin-A receptor antagonist, and sarafotoxin S6c, an endothelin-B receptor agonist.

The estrus cycle, sensitivity to convulsants and the anticonvulsant effect of a neuroactive steroid.

Potentiation of cardiovascular responses to hydralazine by diverse hydrazine derivatives.

Influence of dietary fat on the pharmacodynamics of quinidine, procainamide and tocainide in isolated perfused rabbit hearts.

Pro- and antiarrhythmic effects of d-sotalol and dl-sotalol in an isolated tissue model of ischemia and reperfusion.

Different combinations of retinoids and vitamin D3 analogs efficiently promote growth inhibition and differentiation of myelomonocytic leukemia cell lines.

Establishing benzodiazepines as oral reinforcers: midazolam and diazepam self-administration in rhesus monkeys.

Regulation of [3H]dopamine release from rat striatal slices by sigma receptor ligands.

Ionization and adsorption of a series of local anesthetics in detergent micelles: studies of drug fluorescence.

The bradykinin analog RMP-7 increases intracellular free calcium levels in rat brain microvascular endothelial cells.

The antitumor agent tamoxifen inhibits breakdown of polyphosphoinositides in GH4C1 cells.

Involvement of beta-1 and beta-2 adrenergic receptors in the antidepressant-like effects of centrally administered isoproterenol.

Antagonists of 5-HT4 receptor-mediated responses in adult hippocampal neurons.

Effects of cocaine on the serotonin-induced inward current in rat nodose ganglion neurons.

Effect of the nonpeptide neurotensin antagonist, SR 48692, and two enantiomeric analogs, SR 48527 and SR 49711, on neurotensin binding and contractile responses in guinea pig ileum and colon.

Role of hypogastric nerve activity in opossum internal anal sphincter function: influence of surgical and chemical denervation.

Age modulates the long-term but not the acute effects of the serotonergic neurotoxicant 3,4-methylenedioxymethamphetamine.

Potentiation of lateral hypothalamic and midline mesencephalic brain stimulation reinforcement by nicotine: examination of repeated treatment.

Rate-dependent effects of sematilide on action potential duration in isolated guinea pig ventricular myocytes.

Cocaine interacts with macrophages to modulate mesangial cell proliferation.

Cocaethylene, a metabolite of cocaine and ethanol, is a potent blocker of cardiac sodium channels.

Effect of levcromakalim on hypoxia-, KCl- and prostaglandin F2 alpha-induced contractions in isolated rat pulmonary artery.

Ethanol enhances inward rectification in rat locus ceruleus neurons by increasing the extracellular potassium concentration.

Pharmacological studies with two new ergoline derivatives, the potential antipsychotics LEK-8829 and LEK-8841.

Anxiolytic-like effects of the novel cholinergic channel activator ABT-418.

Modulation of three types of K+ currents in canine coronary artery smooth muscle cells by NS-004, or 1-(2'-hydroxy-5'-chlorophenyl)-5-trifluoromethyl-2(3H) benzimidazolone.

Multiple systems for the biliary excretion of organic anions in rats: liquiritigenin conjugates as model compounds.

5-Hydroxytryptamine-2 and -4 receptors located on bovine isolated mesenteric lymphatics.

A functional beta-2 adrenoceptor-mediated chronotropic response in isolated guinea pig heart tissue: selectivity of the potent beta-2 adrenoceptor agonist TA 2005.

Characterization of dilator prostanoid receptors in the fetal rabbit ductus arteriosus.

Beta-adrenergic regulation of gap-junctional intercellular communication in cultured rabbit gastric epithelial cells.

Loop diuretics affect transcellular electrolyte transport in cells of the distal convoluted tubule.

Induction of heart heme oxygenase-1 (HSP32) by hyperthermia: possible role in stress-mediated elevation of cyclic 3':5'-guanosine monophosphate.

In vitro and in vivo inhibition of rat vascular smooth muscle cell migration and proliferation by a 2-aminochromone U-86983.

Increases in guanine nucleotide binding to striatal G proteins is associated with dopamine receptor supersensitivity.

Angiotensin type 1 receptors mediate smooth muscle proliferation and endothelin biosynthesis in rat vascular smooth muscle.

The 21-aminosteroid tirilazad mesylate protects against endotoxin shock and acute liver failure in rats.

Effects of prostacyclin analogs on the synthesis of tissue factor, tumor necrosis factor-alpha and interleukin-1 beta in human monocytic THP-1 cells.

[125I]iodoproxyfan, a new antagonist to label and visualize cerebral histamine H3 receptors.

Effects of chronic haloperidol and clozapine treatment on neurotensin and c-fos mRNA in rat neostriatal subregions.

Role of thyroid status in the ontogeny of adrenergic cell signaling in rat brain: beta receptors, adenylate cyclase, ornithine decarboxylase and c-fos protooncogene expression.

[3H]RS-23597-190, a potent 5-hydroxytryptamine4 antagonist labels sigma-1 but not sigma-2 binding sites in guinea pig brain.

Diversity of nicotinic acetylcholine receptors in rat hippocampal neurons. II. The rundown and inward rectification of agonist-elicited whole-cell currents and identification of receptor subunits by in situ hybridization.

Bradykinin (Bk) increases cytosolic calcium in cultured rat myenteric neurons via Bk-2 type receptors coupled to mobilization of extracellular and intracellular sources of calcium: evidence that calcium influx is prostaglandin dependent.

Nephrotoxicity and hepatotoxicity of 5,6-dichloro-4-thia-5-hexenoic acid: evidence for fatty acid beta-oxidation-dependent bioactivation.

Intrastriatal Ro15-4513 functionally antagonizes ethanol-induced motor incoordination and striatal adenosinergic modulation of ethanol-induced motor incoordination in rats.

Biochemical and electrophysiological mechanisms of the positive inotropic effect of calyculin A, a protein phosphatase inhibitor.

Adenosine receptors mediate cellular adaptation to ethanol in NG108-15 cells.

Use of midazolam as a human cytochrome P450 3A probe: I. In vitro-in vivo correlations in liver transplant patients.

Use of midazolam as a human cytochrome P450 3A probe: II. Characterization of inter- and intraindividual hepatic CYP3A variability after liver transplantation.

Induction of 12-lipoxygenase expression by epidermal growth factor is mediated by protein kinase C in A431 cells.

EM574, an erythromycin derivative, is a potent motilin receptor agonist in human gastric antrum.

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