Table of Contents

October 1988; 247 (1)

Select this article
- P C Wong,
- A T Chiu,
- W A Price,
- M J Thoolen,
- D J Carini,
- A L Johnson,
- R I Taber,
- and P B Timmermans
Nonpeptide angiotensin II receptor antagonists. I. Pharmacological characterization of 2-n-butyl-4-chloro-1-(2-chlorobenzyl)imidazole-5-acetic acid, sodium salt (S-8307).
J Pharmacol Exp Ther October 1988 247:1-7
- Abstract
- Full Text (PDF)
Select this article
- C P Sung,
- A J Arleth,
- K Shikano,
- and B A Berkowitz
Characterization and function of bradykinin receptors in vascular endothelial cells.
J Pharmacol Exp Ther October 1988 247:8-13
- Abstract
- Full Text (PDF)
Select this article
- L L Devaud and
- T F Murray
Involvement of peripheral-type benzodiazepine receptors in the proconvulsant actions of pyrethroid insecticides.
J Pharmacol Exp Ther October 1988 247:14-22
- Abstract
- Full Text (PDF)
Select this article
- J F French and
- M A Matlib
Identification of a high-affinity peripheral-type benzodiazepine binding site in rat aortic smooth muscle membranes.
J Pharmacol Exp Ther October 1988 247:23-28
- Abstract
- Full Text (PDF)
Select this article
- A D Weissman,
- T P Su,
- J C Hedreen,
- and E D London
Sigma receptors in post-mortem human brains.
J Pharmacol Exp Ther October 1988 247:29-33
- Abstract
- Full Text (PDF)
Select this article
- P J Silver,
- R E Lepore,
- B O'Connor,
- B M Lemp,
- L T Hamel,
- R G Bentley,
- and A L Harris
Inhibition of the low Km cyclic AMP phosphodiesterase and activation of the cyclic AMP system in vascular smooth muscle by milrinone.
J Pharmacol Exp Ther October 1988 247:34-42
- Abstract
- Full Text (PDF)
Select this article
- G J Trachte,
- P J Hook,
- J R Kemp,
- E P Acosta,
- and R J Ziegler
Thromboxane synthesis and actions in isolated adrenergic nerve (pheochromocytoma-12) cells.
J Pharmacol Exp Ther October 1988 247:43-46
- Abstract
- Full Text (PDF)
Select this article
- W K Bickel,
- M L Stitzer,
- G E Bigelow,
- I A Liebson,
- D R Jasinski,
- and R E Johnson
Buprenorphine: dose-related blockade of opioid challenge effects in opioid dependent humans.
J Pharmacol Exp Ther October 1988 247:47-53
- Abstract
- Full Text (PDF)
Select this article
- J D Winkler,
- H M Sarau,
- J J Foley,
- and S T Crooke
Leukotriene D4-induced homologous desensitization in basal and differentiated U-937 cells: characterization with the partial agonist leukotriene E4 and assessment of receptor reserve.
J Pharmacol Exp Ther October 1988 247:54-62
- Abstract
- Full Text (PDF)
Select this article
- J P Pieroni,
- F Dray,
- C R Pace-Asciak,
- and J C McGiff
Identification of 6-keto-prostaglandin E1 obtained from isolated perfused kidney of the rabbit.
J Pharmacol Exp Ther October 1988 247:63-68
- Abstract
- Full Text (PDF)
Select this article
- A L Sirén and
- G Feuerstein
Cardiovascular effects of rat calcitonin gene-related peptide in the conscious rat.
J Pharmacol Exp Ther October 1988 247:69-78
- Abstract
- Full Text (PDF)
Select this article
- D M Stone,
- M Johnson,
- G R Hanson,
- and J W Gibb
Role of endogenous dopamine in the central serotonergic deficits induced by 3,4-methylenedioxymethamphetamine.
J Pharmacol Exp Ther October 1988 247:79-87
- Abstract
- Full Text (PDF)
Select this article
- J K Zubieta,
- E J Cragoe, Jr,
- and L X Cubeddu
Effects of amiloride and 5-(N,N-hexamethylene)amiloride on dopaminergic and cholinergic neurotransmission.
J Pharmacol Exp Ther October 1988 247:88-95
- Abstract
- Full Text (PDF)
Select this article
- E J Zambraski,
- D C Atkinson,
- and J Diamond
Effects of salicylate vs. aspirin on renal prostaglandins and function in normal and sodium-depleted dogs.
J Pharmacol Exp Ther October 1988 247:96-103
- Abstract
- Full Text (PDF)
Select this article
- N Jaiswal,
- G Lambrecht,
- E Mutschler,
- and K U Malik
Contribution of M2 alpha and M2 beta muscarinic receptors to the action of cholinergic stimuli on prostaglandin synthesis and mechanical function in the isolated rabbit heart.
J Pharmacol Exp Ther October 1988 247:104-113
- Abstract
- Full Text (PDF)
Select this article
- S G Oakes,
- P A Iaizzo,
- E Richelson,
- and G Powis
Histamine-induced intracellular free Ca++, inositol phosphates and electrical changes in murine N1E-115 neuroblastoma cells.
J Pharmacol Exp Ther October 1988 247:114-121
- Abstract
- Full Text (PDF)
Select this article
- R N Daly,
- A C Sulpizio,
- B Levitt,
- R M DeMarinis,
- J W Regan,
- R R Ruffolo, Jr,
- and J P Hieble
Evidence for heterogeneity between pre- and postjunctional alpha-2 adrenoceptors using 9-substituted 3-benzazepines.
J Pharmacol Exp Ther October 1988 247:122-128
- Abstract
- Full Text (PDF)
Select this article
- S B Weinberger and
- J L Martinez, Jr
Characterization of hydrolysis of [leu]enkephalin and D-ala2-[L-leu]enkephalin in rat plasma.
J Pharmacol Exp Ther October 1988 247:129-135
- Abstract
- Full Text (PDF)
Select this article
- T Scott and
- K K McMahon
Antagonists and agonists interactions with the muscarinic receptor of the rat large airways.
J Pharmacol Exp Ther October 1988 247:136-142
- Abstract
- Full Text (PDF)
Select this article
- P L Smith,
- G P McCafferty,
- J D Fondacaro,
- M A Wasserman,
- E Elton,
- and F M Ryan
Effects of putative thromboxane receptor agonists and antagonists on rat small intestinal ion transport.
J Pharmacol Exp Ther October 1988 247:143-149
- Abstract
- Full Text (PDF)
Select this article
- U Agnarsson,
- T Tajima,
- and A J Pappano
Carbachol depolarizes and accelerates pacemaker activity in the sinoatrial node of chicks treated with pertussis toxin.
J Pharmacol Exp Ther October 1988 247:150-155
- Abstract
- Full Text (PDF)
Select this article
- J J Liccione and
- M D Maines
Selective vulnerability of glutathione metabolism and cellular defense mechanisms in rat striatum to manganese.
J Pharmacol Exp Ther October 1988 247:156-161
- Abstract
- Full Text (PDF)
Select this article
- G D Olsen,
- T M Cline,
- and K M Sommer
Comparison of chronic morphine and placebo infusion in late gestation fetal lambs: effect upon survival and breathing movements.
J Pharmacol Exp Ther October 1988 247:162-168
- Abstract
- Full Text (PDF)
Select this article
- E Sanders-Bush and
- M Breeding
Putative selective 5-HT-2 antagonists block serotonin 5-HT-1c receptors in the choroid plexus.
J Pharmacol Exp Ther October 1988 247:169-173
- Abstract
- Full Text (PDF)
Select this article
- M W Dudley,
- B W Siegel,
- A M Ogden,
- and D R McCarty
A low dose of xylamine produces sustained and selective decreases in rat brain norepinephrine without evidence of neuronal degeneration.
J Pharmacol Exp Ther October 1988 247:174-179
- Abstract
- Full Text (PDF)
Select this article
- P K Sonsalla,
- L Manzino,
- and R E Heikkila
Interactions of D1 and D2 dopamine receptors on the ipsilateral vs. contralateral side in rats with unilateral lesions of the dopaminergic nigrostriatal pathway.
J Pharmacol Exp Ther October 1988 247:180-185
- Abstract
- Full Text (PDF)
Select this article
- E H Ohlstein,
- L I Kruse,
- M Ezekiel,
- and R N Willette
Further characterization of the cardiovascular effects of the dopamine beta-hydroxylase inhibitor SK&F 102698 in conscious hypertensive rats.
J Pharmacol Exp Ther October 1988 247:186-195
- Abstract
- Full Text (PDF)
Select this article
- G Jagadeesh and
- R C Deth
Phorbol ester-induced modulation of agonist binding to alpha-1 adrenergic receptors in bovine aortic membranes.
J Pharmacol Exp Ther October 1988 247:196-202
- Abstract
- Full Text (PDF)
Select this article
- L J Lee,
- J A Cook,
- and D E Smith
Renal transport kinetics of chlorothiazide in the isolated perfused rat kidney.
J Pharmacol Exp Ther October 1988 247:203-208
- Abstract
- Full Text (PDF)
Select this article
- B J Undem,
- P T Peachell,
- and L M Lichtenstein
Isoproterenol-induced inhibition of immunoglobulin E-mediated release of histamine and arachidonic acid metabolites from the human lung mast cell.
J Pharmacol Exp Ther October 1988 247:209-217
- Abstract
- Full Text (PDF)
Select this article
- J A Warner,
- L M Lichtenstein,
- and D W MacGlashan, Jr
Effects of a specific inhibitor of the 5-lipoxygenase pathway on mediator release from human basophils and mast cells.
J Pharmacol Exp Ther October 1988 247:218-222
- Abstract
- Full Text (PDF)
Select this article
- R K Hester
Functional importance of alpha adrenoceptor-mediated, D600-insensitive Ca++ entry in rabbit aorta.
J Pharmacol Exp Ther October 1988 247:223-234
- Abstract
- Full Text (PDF)
Select this article
- K Inui,
- T Okano,
- H Maegawa,
- M Kato,
- M Takano,
- and R Hori
H+ coupled transport of p.o. cephalosporins via dipeptide carriers in rabbit intestinal brush-border membranes: difference of transport characteristics between cefixime and cephradine.
J Pharmacol Exp Ther October 1988 247:235-241
- Abstract
- Full Text (PDF)
Select this article
- S V Otton,
- H K Crewe,
- M S Lennard,
- G T Tucker,
- and H F Woods
Use of quinidine inhibition to define the role of the sparteine/debrisoquine cytochrome P450 in metoprolol oxidation by human liver microsomes.
J Pharmacol Exp Ther October 1988 247:242-247
- Abstract
- Full Text (PDF)
Select this article
- G Suarez-Kurtz and
- G J Kaczorowski
Effects of dichlorobenzamil on calcium currents in clonal GH3 pituitary cells.
J Pharmacol Exp Ther October 1988 247:248-253
- Abstract
- Full Text (PDF)
Select this article
- V Lagente,
- Z B Fortes,
- J Garcia-Leme,
- and B B Vargaftig
PAF-acether and endotoxin display similar effects on rat mesenteric microvessels: inhibition by specific antagonists.
J Pharmacol Exp Ther October 1988 247:254-261
- Abstract
- Full Text (PDF)
Select this article
- A W Obianime,
- S J Hirst,
- and M M Dale
Interactions between phorbol esters and agents which increase cytosolic calcium in the guinea pig parenchymal strip: direct and indirect effects on the contractile response.
J Pharmacol Exp Ther October 1988 247:262-270
- Abstract
- Full Text (PDF)
Select this article
- D W Rurak,
- S D Yoo,
- E Kwan,
- S M Taylor,
- K W Riggs,
- and J E Axelson
Effects of diphenhydramine in the fetal lamb after maternal or fetal administration.
J Pharmacol Exp Ther October 1988 247:271-278
- Abstract
- Full Text (PDF)
Select this article
- M A Czuba,
- G W Mihaly,
- M S Ching,
- D J Morgan,
- K J Hardy,
- and R A Smallwood
Effects of gestational age on the disposition of propranolol in pregnant sheep.
J Pharmacol Exp Ther October 1988 247:279-282
- Abstract
- Full Text (PDF)
Select this article
- A Mülsch,
- R Busse,
- S Liebau,
- and U Förstermann
LY 83583 interferes with the release of endothelium-derived relaxing factor and inhibits soluble guanylate cyclase.
J Pharmacol Exp Ther October 1988 247:283-288
- Abstract
- Full Text (PDF)
Select this article
- I B Lindén,
- E Nissinen,
- E Etemadzadeh,
- S Kaakkola,
- P Männistö,
- and P Pohto
Favorable effect of catechol-O-methyltransferase inhibition by OR-462 in experimental models of Parkinson's disease.
J Pharmacol Exp Ther October 1988 247:289-293
- Abstract
- Full Text (PDF)
Select this article
- L Beani,
- C Bianchi,
- S Tanganelli,
- T Antonelli,
- M Simonato,
- and S Rando
Inversion of the alpha-2 and alpha-1 noradrenergic control of the cortical release of acetylcholine and gamma-aminobutyric acid in morphine-tolerant guinea pigs.
J Pharmacol Exp Ther October 1988 247:294-301
- Abstract
- Full Text (PDF)
Select this article
- T Katsuragi,
- T Tokunaga,
- K Miyamoto,
- L Kuratomi,
- and T Furukawa
Norepinephrine and adenosine triphosphate release in different ratio from guinea pig vas deferens by high potassium chloride, ouabain and monensin.
J Pharmacol Exp Ther October 1988 247:302-308
- Abstract
- Full Text (PDF)
Select this article
- T Dennis,
- A Dubois,
- J Benavides,
- and B Scatton
Distribution of central omega 1 (benzodiazepine1) and omega 2 (benzodiazepine2) receptor subtypes in the monkey and human brain. An autoradiographic study with [3H]flunitrazepam and the omega 1 selective ligand [3H]zolpidem.
J Pharmacol Exp Ther October 1988 247:309-322
- Abstract
- Full Text (PDF)
Select this article
- S M de Morais and
- P G Wells
Deficiency in bilirubin UDP-glucuronyl transferase as a genetic determinant of acetaminophen toxicity.
J Pharmacol Exp Ther October 1988 247:323-331
- Abstract
- Full Text (PDF)
Select this article
- D Bouhassira,
- L Villanueva,
- and D Le Bars
Intracerebroventricular morphine decreases descending inhibitions acting on lumbar dorsal horn neuronal activities related to pain in the rat.
J Pharmacol Exp Ther October 1988 247:332-342
- Abstract
- Full Text (PDF)
Select this article
- K J Nicklaus,
- P McGonigle,
- and P B Molinoff
[3H]SCH 23390 labels both dopamine-1 and 5-hydroxytryptamine1c receptors in the choroid plexus.
J Pharmacol Exp Ther October 1988 247:343-348
- Abstract
- Full Text (PDF)
Select this article
- P D Holohan,
- P P Sokol,
- C R Ross,
- R Coulson,
- M E Trimble,
- D A Laska,
- and P D Williams
Gentamicin-induced increases in cytosolic calcium in pig kidney cells (LLC-PK1).
J Pharmacol Exp Ther October 1988 247:349-354
- Abstract
- Full Text (PDF)
Select this article
- R F Cox,
- J L Neumeyer,
- and B L Waszczak
Effects of N-n-propylnorapomorphine enantiomers on single unit activity of substantia nigra pars compacta and ventral tegmental area dopamine neurons.
J Pharmacol Exp Ther October 1988 247:355-362
- Abstract
- Full Text (PDF)
Select this article
- G Matera,
- J A Cook,
- R A Hennigar,
- G E Tempel,
- W C Wise,
- T D Oglesby,
- and P V Halushka
Beneficial effects of a 5-lipoxygenase inhibitor in endotoxic shock in the rat.
J Pharmacol Exp Ther October 1988 247:363-371
- Abstract
- Full Text (PDF)
Select this article
- D J Hinman and
- H H Szeto
Cholinergic influences on sleep-wake patterns and breathing movements in the fetus.
J Pharmacol Exp Ther October 1988 247:372-378
- Abstract
- Full Text (PDF)
Select this article
- G A Ordway,
- C Gambarana,
- and A Frazer
Quantitative autoradiography of central beta adrenoceptor subtypes: comparison of the effects of chronic treatment with desipramine or centrally administered l-isoproterenol.
J Pharmacol Exp Ther October 1988 247:379-389
- Abstract
- Full Text (PDF)
Select this article
- N Mahy,
- M Woolkalis,
- D Manning,
- and T Reisine
Characteristics of somatostatin desensitization in the pituitary tumor cell line AtT-20.
J Pharmacol Exp Ther October 1988 247:390-396
- Abstract
- Full Text (PDF)

Article

Select this article

ERRATUM
J Pharmacol Exp Ther October 1988 247:397
- Abstract
- Full Text (PDF)

Current Issue

November 2009, 331 (2)

Nonpeptide angiotensin II receptor antagonists. I. Pharmacological characterization of 2-n-butyl-4-chloro-1-(2-chlorobenzyl)imidazole-5-acetic acid, sodium salt (S-8307).

Characterization and function of bradykinin receptors in vascular endothelial cells.

Involvement of peripheral-type benzodiazepine receptors in the proconvulsant actions of pyrethroid insecticides.

Identification of a high-affinity peripheral-type benzodiazepine binding site in rat aortic smooth muscle membranes.

Sigma receptors in post-mortem human brains.

Inhibition of the low Km cyclic AMP phosphodiesterase and activation of the cyclic AMP system in vascular smooth muscle by milrinone.

Thromboxane synthesis and actions in isolated adrenergic nerve (pheochromocytoma-12) cells.

Buprenorphine: dose-related blockade of opioid challenge effects in opioid dependent humans.

Leukotriene D4-induced homologous desensitization in basal and differentiated U-937 cells: characterization with the partial agonist leukotriene E4 and assessment of receptor reserve.

Identification of 6-keto-prostaglandin E1 obtained from isolated perfused kidney of the rabbit.

Cardiovascular effects of rat calcitonin gene-related peptide in the conscious rat.

Role of endogenous dopamine in the central serotonergic deficits induced by 3,4-methylenedioxymethamphetamine.

Effects of amiloride and 5-(N,N-hexamethylene)amiloride on dopaminergic and cholinergic neurotransmission.

Effects of salicylate vs. aspirin on renal prostaglandins and function in normal and sodium-depleted dogs.

Contribution of M2 alpha and M2 beta muscarinic receptors to the action of cholinergic stimuli on prostaglandin synthesis and mechanical function in the isolated rabbit heart.

Histamine-induced intracellular free Ca++, inositol phosphates and electrical changes in murine N1E-115 neuroblastoma cells.

Evidence for heterogeneity between pre- and postjunctional alpha-2 adrenoceptors using 9-substituted 3-benzazepines.

Characterization of hydrolysis of [leu]enkephalin and D-ala2-[L-leu]enkephalin in rat plasma.

Antagonists and agonists interactions with the muscarinic receptor of the rat large airways.

Effects of putative thromboxane receptor agonists and antagonists on rat small intestinal ion transport.

Carbachol depolarizes and accelerates pacemaker activity in the sinoatrial node of chicks treated with pertussis toxin.

Selective vulnerability of glutathione metabolism and cellular defense mechanisms in rat striatum to manganese.

Comparison of chronic morphine and placebo infusion in late gestation fetal lambs: effect upon survival and breathing movements.

Putative selective 5-HT-2 antagonists block serotonin 5-HT-1c receptors in the choroid plexus.

A low dose of xylamine produces sustained and selective decreases in rat brain norepinephrine without evidence of neuronal degeneration.

Interactions of D1 and D2 dopamine receptors on the ipsilateral vs. contralateral side in rats with unilateral lesions of the dopaminergic nigrostriatal pathway.

Further characterization of the cardiovascular effects of the dopamine beta-hydroxylase inhibitor SK&F 102698 in conscious hypertensive rats.

Phorbol ester-induced modulation of agonist binding to alpha-1 adrenergic receptors in bovine aortic membranes.

Renal transport kinetics of chlorothiazide in the isolated perfused rat kidney.

Isoproterenol-induced inhibition of immunoglobulin E-mediated release of histamine and arachidonic acid metabolites from the human lung mast cell.

Effects of a specific inhibitor of the 5-lipoxygenase pathway on mediator release from human basophils and mast cells.

Functional importance of alpha adrenoceptor-mediated, D600-insensitive Ca++ entry in rabbit aorta.

H+ coupled transport of p.o. cephalosporins via dipeptide carriers in rabbit intestinal brush-border membranes: difference of transport characteristics between cefixime and cephradine.

Use of quinidine inhibition to define the role of the sparteine/debrisoquine cytochrome P450 in metoprolol oxidation by human liver microsomes.

Effects of dichlorobenzamil on calcium currents in clonal GH3 pituitary cells.

PAF-acether and endotoxin display similar effects on rat mesenteric microvessels: inhibition by specific antagonists.

Interactions between phorbol esters and agents which increase cytosolic calcium in the guinea pig parenchymal strip: direct and indirect effects on the contractile response.

Effects of diphenhydramine in the fetal lamb after maternal or fetal administration.

Effects of gestational age on the disposition of propranolol in pregnant sheep.

LY 83583 interferes with the release of endothelium-derived relaxing factor and inhibits soluble guanylate cyclase.

Favorable effect of catechol-O-methyltransferase inhibition by OR-462 in experimental models of Parkinson's disease.

Inversion of the alpha-2 and alpha-1 noradrenergic control of the cortical release of acetylcholine and gamma-aminobutyric acid in morphine-tolerant guinea pigs.

Norepinephrine and adenosine triphosphate release in different ratio from guinea pig vas deferens by high potassium chloride, ouabain and monensin.

Distribution of central omega 1 (benzodiazepine1) and omega 2 (benzodiazepine2) receptor subtypes in the monkey and human brain. An autoradiographic study with [3H]flunitrazepam and the omega 1 selective ligand [3H]zolpidem.

Deficiency in bilirubin UDP-glucuronyl transferase as a genetic determinant of acetaminophen toxicity.

Intracerebroventricular morphine decreases descending inhibitions acting on lumbar dorsal horn neuronal activities related to pain in the rat.

[3H]SCH 23390 labels both dopamine-1 and 5-hydroxytryptamine1c receptors in the choroid plexus.

Gentamicin-induced increases in cytosolic calcium in pig kidney cells (LLC-PK1).

Effects of N-n-propylnorapomorphine enantiomers on single unit activity of substantia nigra pars compacta and ventral tegmental area dopamine neurons.

Beneficial effects of a 5-lipoxygenase inhibitor in endotoxic shock in the rat.

Cholinergic influences on sleep-wake patterns and breathing movements in the fetus.

Quantitative autoradiography of central beta adrenoceptor subtypes: comparison of the effects of chronic treatment with desipramine or centrally administered l-isoproterenol.

Characteristics of somatostatin desensitization in the pituitary tumor cell line AtT-20.

Article

ERRATUM

This Issue

Current Issue