Table of Contents

May 1987; 241 (2)

Select this article
- N A Flavahan,
- J P Cooke,
- J T Shepherd,
- and P M Vanhoutte
Human postjunctional alpha-1 and alpha-2 adrenoceptors: differential distribution in arteries of the limbs.
J Pharmacol Exp Ther May 1987 241:361-365
- Abstract
- Full Text (PDF)
Select this article
- W S Lai and
- E E el-Fakahany
Phorbol ester-induced inhibition of cyclic GMP formation mediated by muscarinic receptors in murine neuroblastoma cells.
J Pharmacol Exp Ther May 1987 241:366-373
- Abstract
- Full Text (PDF)
Select this article
- D M Zimmerman,
- J D Leander,
- J K Reel,
- and M D Hynes
Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.
J Pharmacol Exp Ther May 1987 241:374-378
- Abstract
- Full Text (PDF)
Select this article
- J S Williams,
- Y H Baik,
- W J Koch,
- and A Schwartz
A possible role for the endothelium in porcine coronary smooth muscle responses to dihydropyridine calcium channel modulators.
J Pharmacol Exp Ther May 1987 241:379-386
- Abstract
- Full Text (PDF)
Select this article
- M R Hynes and
- S P Duckles
Effect of increasing age on the endothelium-mediated relaxation of rat blood vessels in vitro.
J Pharmacol Exp Ther May 1987 241:387-392
- Abstract
- Full Text (PDF)
Select this article
- F Porreca,
- J S Heyman,
- H I Mosberg,
- J R Omnaas,
- and J L Vaught
Role of mu and delta receptors in the supraspinal and spinal analgesic effects of [D-Pen2, D-Pen5]enkephalin in the mouse.
J Pharmacol Exp Ther May 1987 241:393-400
- Abstract
- Full Text (PDF)
Select this article
- S Kawai,
- L K Nieman,
- D D Brandon,
- R Udelsman,
- D L Loriaux,
- and G P Chrousos
Pharmacokinetic properties of the antiglucocorticoid and antiprogesterone steroid RU 486 in man.
J Pharmacol Exp Ther May 1987 241:401-406
- Abstract
- Full Text (PDF)
Select this article
- M K Ahlijanian and
- D M Cooper
Antagonism of calmodulin-stimulated adenylate cyclase by trifluoperazine, calmidazolium and W-7 in rat cerebellar membranes.
J Pharmacol Exp Ther May 1987 241:407-414
- Abstract
- Full Text (PDF)
Select this article
- M Williams,
- J Francis,
- G Ghai,
- A Braunwalder,
- S Psychoyos,
- G A Stone,
- and W D Cash
Biochemical characterization of the triazoloquinazoline, CGS 15943, a novel, non-xanthine adenosine antagonist.
J Pharmacol Exp Ther May 1987 241:415-420
- Abstract
- Full Text (PDF)
Select this article
- W Balduini,
- S D Murphy,
- and L G Costa
Developmental changes in muscarinic receptor-stimulated phosphoinositide metabolism in rat brain.
J Pharmacol Exp Ther May 1987 241:421-427
- Abstract
- Full Text (PDF)
Select this article
- R J McGonigle,
- J Brookins,
- B L Pegram,
- and J W Fisher
Enhanced erythropoietin production by calcium entry blockers in rats exposed to hypoxia.
J Pharmacol Exp Ther May 1987 241:428-432
- Abstract
- Full Text (PDF)
Select this article
- R J Wills,
- H E Gallo-Torres,
- R Bertko,
- and B H Min
Pharmacokinetics and antisecretory activity of trimoprostil in Heidenhain-pouch dogs.
J Pharmacol Exp Ther May 1987 241:433-437
- Abstract
- Full Text (PDF)
Select this article
- B M Sharp,
- H S Beyer,
- A S Levine,
- J E Morley,
- and K M McAllen
Attenuation of the plasma prolactin response to restraint stress after acute and chronic administration of nicotine to rats.
J Pharmacol Exp Ther May 1987 241:438-442
- Abstract
- Full Text (PDF)
Select this article
- A A Letter,
- K Merchant,
- J W Gibb,
- and G R Hanson
Effect of methamphetamine on neurotensin concentrations in rat brain regions.
J Pharmacol Exp Ther May 1987 241:443-447
- Abstract
- Full Text (PDF)
Select this article
- S Sabatini,
- W C Yang,
- and N A Kurtzman
Effect of parathyroid hormone fragments on calcium transport in toad bladder.
J Pharmacol Exp Ther May 1987 241:448-452
- Abstract
- Full Text (PDF)
Select this article
- M H Hawthorn,
- D A Taylor,
- and W W Fleming
Characteristics of adaptive supersensitivity in the left atrium of the guinea pig.
J Pharmacol Exp Ther May 1987 241:453-457
- Abstract
- Full Text (PDF)
Select this article
- P F Wick,
- A C Keung,
- J J Bowler,
- and R C Deth
Alpha-1 adrenergic coupling events induced by full and partial agonists in rabbit aorta.
J Pharmacol Exp Ther May 1987 241:458-464
- Abstract
- Full Text (PDF)
Select this article
- D W Pomfret,
- K W Schenck,
- P Fludzinski,
- and M L Cohen
Interaction of 5-hydroxykynurenamine, L-kynurenine and kynuramine with multiple serotonin receptors in smooth muscle.
J Pharmacol Exp Ther May 1987 241:465-471
- Abstract
- Full Text (PDF)
Select this article
- D W Wolff,
- F A Gesek,
- and J W Strandhoy
In vivo assessment of rat renal alpha adrenoceptors.
J Pharmacol Exp Ther May 1987 241:472-476
- Abstract
- Full Text (PDF)
Select this article
- J K Belknap,
- P W Danielson,
- S E Laursen,
- and B Noordewier
Selective breeding for levorphanol-induced antinociception on the hot-plate assay: commonalities in mechanism of action with morphine, pentazocine, ethylketocyclazocine, U-50488H and clonidine in mice.
J Pharmacol Exp Ther May 1987 241:477-481
- Abstract
- Full Text (PDF)
Select this article
- J Kao and
- J Hall
Skin absorption and cutaneous first pass metabolism of topical steroids: in vitro studies with mouse skin in organ culture.
J Pharmacol Exp Ther May 1987 241:482-487
- Abstract
- Full Text (PDF)
Select this article
- R E Vestal,
- B J Cusack,
- G D Mercer,
- G W Dawson,
- and B K Park
Aging and drug interactions. I. Effect of cimetidine and smoking on the oxidation of theophylline and cortisol in healthy men.
J Pharmacol Exp Ther May 1987 241:488-500
- Abstract
- Full Text (PDF)
Select this article
- D A Houston,
- G Burnstock,
- and P M Vanhoutte
Different P2-purinergic receptor subtypes of endothelium and smooth muscle in canine blood vessels.
J Pharmacol Exp Ther May 1987 241:501-506
- Abstract
- Full Text (PDF)
Select this article
- D C Rees,
- J S Knisely,
- R L Balster,
- S Jordan,
- and T J Breen
Pentobarbital-like discriminative stimulus properties of halothane, 1,1,1-trichloroethane, isoamyl nitrite, flurothyl and oxazepam in mice.
J Pharmacol Exp Ther May 1987 241:507-515
- Abstract
- Full Text (PDF)
Select this article
- P D Cherry and
- C N Gillis
Evidence for the role of endothelium-derived relaxing factor in acetylcholine-induced vasodilatation in the intact lung.
J Pharmacol Exp Ther May 1987 241:516-520
- Abstract
- Full Text (PDF)
Select this article
- P M Beardsley,
- J A Scimeca,
- and B R Martin
Studies on the agonistic activity of delta 9-11-tetrahydrocannabinol in mice, dogs and rhesus monkeys and its interactions with delta 9-tetrahydrocannabinol.
J Pharmacol Exp Ther May 1987 241:521-526
- Abstract
- Full Text (PDF)
Select this article
- D W Roberts,
- N R Pumford,
- D W Potter,
- R W Benson,
- and J A Hinson
A sensitive immunochemical assay for acetaminophen-protein adducts.
J Pharmacol Exp Ther May 1987 241:527-533
- Abstract
- Full Text (PDF)
Select this article
- P J Vaysse,
- E L Gardner,
- and R S Zukin
Modulation of rat brain opioid receptors by cannabinoids.
J Pharmacol Exp Ther May 1987 241:534-539
- Abstract
- Full Text (PDF)
Select this article
- J A Gondal,
- J L Eiseman,
- and A P Alvares
Regulation of heme metabolism and monooxygeneses in liver and kidney: influence of therapeutically used gold compounds.
J Pharmacol Exp Ther May 1987 241:540-546
- Abstract
- Full Text (PDF)
Select this article
- G Eisenhofer,
- T G Ropchak,
- R W Stull,
- D S Goldstein,
- H R Keiser,
- and I J Kopin
Dihydroxyphenylglycol and intraneuronal metabolism of endogenous and exogenous norepinephrine in the rat vas deferens.
J Pharmacol Exp Ther May 1987 241:547-553
- Abstract
- Full Text (PDF)
Select this article
- E H Ohlstein,
- L I Kruse,
- M Ezekiel,
- S S Sherman,
- R Erickson,
- W E DeWolf, Jr,
- and B A Berkowitz
Cardiovascular effects of a new potent dopamine beta-hydroxylase inhibitor in spontaneously hypertensive rats.
J Pharmacol Exp Ther May 1987 241:554-559
- Abstract
- Full Text (PDF)
Select this article
- M Chiariello,
- G Ambrosio,
- M Cappelli-Bigazzi,
- E Nevola,
- P Perrone-Filardi,
- G Marone,
- and M Condorelli
Inhibition of ischemia-induced phospholipase activation by quinacrine protects jeopardized myocardium in rats with coronary artery occlusion.
J Pharmacol Exp Ther May 1987 241:560-568
- Abstract
- Full Text (PDF)
Select this article
- G L Kovács,
- Z Sarnyai,
- F Izbéki,
- G Szabó,
- G Telegdy,
- T Barth,
- K Jost,
- and F Brtnik
Effects of oxytocin-related peptides on acute morphine tolerance: opposite actions by oxytocin and its receptor antagonists.
J Pharmacol Exp Ther May 1987 241:569-574
- Abstract
- Full Text (PDF)
Select this article
- H Komulainen and
- S C Bondy
Modulation of levels of free calcium within synaptosomes by organochlorine insecticides.
J Pharmacol Exp Ther May 1987 241:575-581
- Abstract
- Full Text (PDF)
Select this article
- M Nishibori,
- Y Itoh,
- R Oishi,
- and K Saeki
Mechanism of the central hyperglycemic action of histamine in mice.
J Pharmacol Exp Ther May 1987 241:582-586
- Abstract
- Full Text (PDF)
Select this article
- K Ishii and
- R Kato
Suppression by muscarinic M2 stimulation of the contractile mechanism via histamine H1 receptors in the longitudinal muscle of guinea pig ileum.
J Pharmacol Exp Ther May 1987 241:587-593
- Abstract
- Full Text (PDF)
Select this article
- A Tsuji,
- T Terasaki,
- I Tamai,
- and H Hirooka
H+ gradient-dependent and carrier-mediated transport of cefixime, a new cephalosporin antibiotic, across brush-border membrane vesicles from rat small intestine.
J Pharmacol Exp Ther May 1987 241:594-601
- Abstract
- Full Text (PDF)
Select this article
- M Tariq,
- N S Parmar,
- and A M Ageel
Gastric and duodenal antiulcer and cytoprotective effects of proglumide in rats.
J Pharmacol Exp Ther May 1987 241:602-607
- Abstract
- Full Text (PDF)
Select this article
- I Llona,
- R Vavrek,
- J Stewart,
- and J P Huidobro-Toro
Identification of pre- and postsynaptic bradykinin receptor sites in the vas deferens: evidence for different structural prerequisites.
J Pharmacol Exp Ther May 1987 241:608-614
- Abstract
- Full Text (PDF)
Select this article
- S Fritz,
- W Lindner,
- I Roots,
- B M Frey,
- and A Küpfer
Stereochemistry of aromatic phenytoin hydroxylation in various drug hydroxylation phenotypes in humans.
J Pharmacol Exp Ther May 1987 241:615-622
- Abstract
- Full Text (PDF)
Select this article
- M Hatmi,
- A del Maschio,
- J Lefort,
- G de gaetano,
- B B Vargaftig,
- and C Cerletti
Effects of sulfinpyrazone and its metabolite G25671 on platelet activation and desensitization and on bronchoconstriction induced by the prostaglandin endoperoxide analog U46619.
J Pharmacol Exp Ther May 1987 241:623-627
- Abstract
- Full Text (PDF)
Select this article
- R Micheletti,
- E Montagna,
- and A Giachetti
AF-DX 116, a cardioselective muscarinic antagonist.
J Pharmacol Exp Ther May 1987 241:628-634
- Abstract
- Full Text (PDF)
Select this article
- K Goto,
- S Kimura,
- and A Saito
Inhibitory effect of calcitonin gene-related peptide on excitation and contraction of smooth muscles of the rat vas deferens.
J Pharmacol Exp Ther May 1987 241:635-641
- Abstract
- Full Text (PDF)
Select this article
- T Dennis,
- R L'Heureux,
- C Carter,
- and B Scatton
Presynaptic alpha-2 adrenoceptors play a major role in the effects of idazoxan on cortical noradrenaline release (as measured by in vivo dialysis) in the rat.
J Pharmacol Exp Ther May 1987 241:642-649
- Abstract
- Full Text (PDF)
Select this article
- T Tsubomura,
- T Okamoto,
- K Kurahashi,
- and M Fujiwara
Gastric excitation by stimulation of the vagal trunk after chronic supranodose vagotomy in cats.
J Pharmacol Exp Ther May 1987 241:650-654
- Abstract
- Full Text (PDF)
Select this article
- M R Mark
Amino acid uptake in denervated rat parotid gland: I. Preparation and evaluation of a lobule system for in vitro studies.
J Pharmacol Exp Ther May 1987 241:655-662
- Abstract
- Full Text (PDF)
Select this article
- M R Mark
Amino acid uptake in the rat parotid gland: II. Effects of surgical sympathectomy and parasympathectomy.
J Pharmacol Exp Ther May 1987 241:663-668
- Abstract
- Full Text (PDF)
Select this article
- S I Harik,
- J W Schmidley,
- L A Iacofano,
- P Blue,
- P K Arora,
- and L M Sayre
On the mechanisms underlying 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine neurotoxicity: the effect of perinigral infusion of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine, its metabolite and their analogs in the rat.
J Pharmacol Exp Ther May 1987 241:669-676
- Abstract
- Full Text (PDF)
Select this article
- J S Yang and
- R W Olsen
gamma-Aminobutyric acid receptor-regulated 36Cl- flux in mouse cortical slices.
J Pharmacol Exp Ther May 1987 241:677-685
- Abstract
- Full Text (PDF)
Select this article
- P A Talbot
Potentiation of aminoglycoside-induced neuromuscular blockade by protons in vitro and in vivo.
J Pharmacol Exp Ther May 1987 241:686-694
- Abstract
- Full Text (PDF)
Select this article
- M E Spearman,
- R M Goodwin,
- L D Apelgren,
- and T F Bumol
Disposition of the monoclonal antibody-vinca alkaloid conjugate KS1/4-DAVLB (LY256787) and free 4-desacetylvinblastine in tumor-bearing nude mice.
J Pharmacol Exp Ther May 1987 241:695-703
- Abstract
- Full Text (PDF)
Select this article
- W A Geary, 2nd,
- G F Wooten,
- J B Perlin,
- and E W Lothman
In vitro and in vivo distribution and binding of phenytoin to rat brain.
J Pharmacol Exp Ther May 1987 241:704-713
- Abstract
- Full Text (PDF)
Select this article
- G A Gerhardt,
- K Pang,
- and G M Rose
In vivo electrochemical demonstration of the presynaptic actions of phencyclidine in rat caudate nucleus.
J Pharmacol Exp Ther May 1987 241:714-721
- Abstract
- Full Text (PDF)
Select this article
- J P Fabisiak,
- E S Vesell,
- and D E Rannels
Interactions of beta adrenergic antagonists with isolated rat alveolar type II pneumocytes. I. Analysis, characterization and regulation of specific beta adrenergic receptors.
J Pharmacol Exp Ther May 1987 241:722-727
- Abstract
- Full Text (PDF)
Select this article
- J P Fabisiak,
- E S Vesell,
- and D E Rannels
Interactions of beta adrenergic antagonists with isolated rat alveolar type II pneumocytes. II. Receptor-independent accumulation of beta adrenergic antagonists and other cationic amphiphilic drugs in lamellar bodies.
J Pharmacol Exp Ther May 1987 241:728-735
- Abstract
- Full Text (PDF)
Select this article
- R B McCall and
- L T Harris
Characterization of the central sympathoinhibitory action of ketanserin.
J Pharmacol Exp Ther May 1987 241:736-740
- Abstract
- Full Text (PDF)
Select this article
- J J Lynch,
- S D Nelson,
- S A MacEwen,
- E M Driscoll,
- and B R Lucchesi
Antifibrillatory efficacy of concomitant beta adrenergic receptor blockade with dilevalol, the R,R-isomer of labetalol, and muscarinic receptor blockade with methylscopolamine.
J Pharmacol Exp Ther May 1987 241:741-749
- Abstract
- Full Text (PDF)

Current Issue

November 2009, 331 (2)

Human postjunctional alpha-1 and alpha-2 adrenoceptors: differential distribution in arteries of the limbs.

Phorbol ester-induced inhibition of cyclic GMP formation mediated by muscarinic receptors in murine neuroblastoma cells.

Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.

A possible role for the endothelium in porcine coronary smooth muscle responses to dihydropyridine calcium channel modulators.

Effect of increasing age on the endothelium-mediated relaxation of rat blood vessels in vitro.

Role of mu and delta receptors in the supraspinal and spinal analgesic effects of [D-Pen2, D-Pen5]enkephalin in the mouse.

Pharmacokinetic properties of the antiglucocorticoid and antiprogesterone steroid RU 486 in man.

Antagonism of calmodulin-stimulated adenylate cyclase by trifluoperazine, calmidazolium and W-7 in rat cerebellar membranes.

Biochemical characterization of the triazoloquinazoline, CGS 15943, a novel, non-xanthine adenosine antagonist.

Developmental changes in muscarinic receptor-stimulated phosphoinositide metabolism in rat brain.

Enhanced erythropoietin production by calcium entry blockers in rats exposed to hypoxia.

Pharmacokinetics and antisecretory activity of trimoprostil in Heidenhain-pouch dogs.

Attenuation of the plasma prolactin response to restraint stress after acute and chronic administration of nicotine to rats.

Effect of methamphetamine on neurotensin concentrations in rat brain regions.

Effect of parathyroid hormone fragments on calcium transport in toad bladder.

Characteristics of adaptive supersensitivity in the left atrium of the guinea pig.

Alpha-1 adrenergic coupling events induced by full and partial agonists in rabbit aorta.

Interaction of 5-hydroxykynurenamine, L-kynurenine and kynuramine with multiple serotonin receptors in smooth muscle.

In vivo assessment of rat renal alpha adrenoceptors.

Selective breeding for levorphanol-induced antinociception on the hot-plate assay: commonalities in mechanism of action with morphine, pentazocine, ethylketocyclazocine, U-50488H and clonidine in mice.

Skin absorption and cutaneous first pass metabolism of topical steroids: in vitro studies with mouse skin in organ culture.

Aging and drug interactions. I. Effect of cimetidine and smoking on the oxidation of theophylline and cortisol in healthy men.

Different P2-purinergic receptor subtypes of endothelium and smooth muscle in canine blood vessels.

Pentobarbital-like discriminative stimulus properties of halothane, 1,1,1-trichloroethane, isoamyl nitrite, flurothyl and oxazepam in mice.

Evidence for the role of endothelium-derived relaxing factor in acetylcholine-induced vasodilatation in the intact lung.

Studies on the agonistic activity of delta 9-11-tetrahydrocannabinol in mice, dogs and rhesus monkeys and its interactions with delta 9-tetrahydrocannabinol.

A sensitive immunochemical assay for acetaminophen-protein adducts.

Modulation of rat brain opioid receptors by cannabinoids.

Regulation of heme metabolism and monooxygeneses in liver and kidney: influence of therapeutically used gold compounds.

Dihydroxyphenylglycol and intraneuronal metabolism of endogenous and exogenous norepinephrine in the rat vas deferens.

Cardiovascular effects of a new potent dopamine beta-hydroxylase inhibitor in spontaneously hypertensive rats.

Inhibition of ischemia-induced phospholipase activation by quinacrine protects jeopardized myocardium in rats with coronary artery occlusion.

Effects of oxytocin-related peptides on acute morphine tolerance: opposite actions by oxytocin and its receptor antagonists.

Modulation of levels of free calcium within synaptosomes by organochlorine insecticides.

Mechanism of the central hyperglycemic action of histamine in mice.

Suppression by muscarinic M2 stimulation of the contractile mechanism via histamine H1 receptors in the longitudinal muscle of guinea pig ileum.

H+ gradient-dependent and carrier-mediated transport of cefixime, a new cephalosporin antibiotic, across brush-border membrane vesicles from rat small intestine.

Gastric and duodenal antiulcer and cytoprotective effects of proglumide in rats.

Identification of pre- and postsynaptic bradykinin receptor sites in the vas deferens: evidence for different structural prerequisites.

Stereochemistry of aromatic phenytoin hydroxylation in various drug hydroxylation phenotypes in humans.

Effects of sulfinpyrazone and its metabolite G25671 on platelet activation and desensitization and on bronchoconstriction induced by the prostaglandin endoperoxide analog U46619.

AF-DX 116, a cardioselective muscarinic antagonist.

Inhibitory effect of calcitonin gene-related peptide on excitation and contraction of smooth muscles of the rat vas deferens.

Presynaptic alpha-2 adrenoceptors play a major role in the effects of idazoxan on cortical noradrenaline release (as measured by in vivo dialysis) in the rat.

Gastric excitation by stimulation of the vagal trunk after chronic supranodose vagotomy in cats.

Amino acid uptake in denervated rat parotid gland: I. Preparation and evaluation of a lobule system for in vitro studies.

Amino acid uptake in the rat parotid gland: II. Effects of surgical sympathectomy and parasympathectomy.

On the mechanisms underlying 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine neurotoxicity: the effect of perinigral infusion of 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine, its metabolite and their analogs in the rat.

gamma-Aminobutyric acid receptor-regulated 36Cl- flux in mouse cortical slices.

Potentiation of aminoglycoside-induced neuromuscular blockade by protons in vitro and in vivo.

Disposition of the monoclonal antibody-vinca alkaloid conjugate KS1/4-DAVLB (LY256787) and free 4-desacetylvinblastine in tumor-bearing nude mice.

In vitro and in vivo distribution and binding of phenytoin to rat brain.

In vivo electrochemical demonstration of the presynaptic actions of phencyclidine in rat caudate nucleus.

Interactions of beta adrenergic antagonists with isolated rat alveolar type II pneumocytes. I. Analysis, characterization and regulation of specific beta adrenergic receptors.

Interactions of beta adrenergic antagonists with isolated rat alveolar type II pneumocytes. II. Receptor-independent accumulation of beta adrenergic antagonists and other cationic amphiphilic drugs in lamellar bodies.

Characterization of the central sympathoinhibitory action of ketanserin.

Antifibrillatory efficacy of concomitant beta adrenergic receptor blockade with dilevalol, the R,R-isomer of labetalol, and muscarinic receptor blockade with methylscopolamine.

This Issue

Current Issue